Browse by Uncontrolled Keywords
Number of items: 18.
2007
Blackie, MAL;
Beagley, P;
Croft, SL;
Kendrick, H;
Moss, JR;
Chibale, K;
(2007)
Metallocene-based antimalarials: An exploration into the influence of the ferrocenyl moiety on in vitro antimalarial activity in chloroquine-sensitive and chloroquine-resistant strains of Plasmodium falciparum.
Bioorganic & medicinal chemistry, 15 (20).
pp. 6510-6516.
ISSN 0968-0896
DOI: https://doi.org/10.1016/j.bmc.2007.07.012
Full text not available from this repository.
Musonda, CC;
Little, S;
Yardley, V;
Chibale, K;
(2007)
Application of multicomponent reactions to antimalarial drug discovery. Part 3: Discovery of aminoxazole 4-aminoquinolines with potent antiplasmodial activity in vitro.
Bioorganic & medicinal chemistry letters, 17 (17).
pp. 4733-4736.
ISSN 0960-894X
DOI: https://doi.org/10.1016/j.bmcl.2007.06.070
Full text not available from this repository.
Too, K;
Brown, DM;
Bongard, E;
Yardley, V;
Vivas, L;
Loakes, D;
(2007)
Anti-malarial activity of N-6-modified purine analogues.
Bioorganic & medicinal chemistry, 15 (16).
pp. 5551-5562.
ISSN 0968-0896
DOI: https://doi.org/10.1016/j.bmc.2007.05.038
Full text not available from this repository.
2006
Hudock, MP;
Sanz-Rodriguez, CE;
Song, YC;
Chan, JMW;
Zhang, YH;
Odeh, S;
Kosztowski, T;
Leon-Rossell, A;
Concepcion, JL;
Yardley, V;
+3 more...
Croft, SL;
Urbina, JA;
Oldfield, E;
(2006)
Inhibition of Trypanosoma cruzi hexokinase by bisphosphonates.
Journal of medicinal chemistry, 49 (1).
pp. 215-223.
ISSN 0022-2623
DOI: https://doi.org/10.1021/jm0582625
Full text not available from this repository.
2005
Lorente, SO;
Jimenez, CJ;
Gros, L;
Yardley, V;
de Luca-Fradley, K;
Croft, SL;
Urbina, JA;
Ruiz-Perez, LM;
Pacanowska, DG;
Gilbert, IH;
(2005)
Preparation of transition-state analogues of sterol 24-methyl transferase as potential anti-parasities.
Bioorganic & medicinal chemistry, 13 (18).
pp. 5435-5453.
ISSN 0968-0896
DOI: https://doi.org/10.1016/j.bmc.2005.06.012
Full text not available from this repository.
2004
Ghosh, S;
Chan, JMW;
Lea, CR;
Meints, GA;
Lewis, JC;
Tovian, ZS;
Flessner, RM;
Loftus, TC;
Bruchhaus, I;
Kendrick, H;
+5 more...
Croft, SL;
Kemp, RG;
Kobayashi, S;
Nozaki, T;
Oldfield, E;
(2004)
Effects of bisphosphonates on the growth of Entamoeba histolytica and Plasmodium species in vitro and in vivo.
Journal of medicinal chemistry, 47 (1).
pp. 175-187.
ISSN 0022-2623
DOI: https://doi.org/10.1021/jm030084x
Full text not available from this repository.
2003
Chauviere, G;
Bouteille, B;
Enanga, B;
de Albuquerque, C;
Croft, SL;
Dumas, M;
Perie, J;
(2003)
Synthesis and biological activity of nitro heterocycles analogous to megazol, a trypanocidal lead.
Journal of medicinal chemistry, 46 (3).
pp. 427-440.
ISSN 0022-2623
DOI: https://doi.org/10.1021/jm021030a
Full text not available from this repository.
Croft, SL;
Seifert, K;
Duchene, M;
(2003)
Antiprotozoal activities of phospholipid analogues.
Molecular and biochemical parasitology, 126 (2).
pp. 165-72.
ISSN 0166-6851
DOI: https://doi.org/10.1016/S0166-6851(02)00283-9
Full text not available from this repository.
Magaraci, F;
Jimenez, CJ;
Rodrigues, C;
Rodrigues, JCF;
Braga, MV;
Yardley, V;
de Luca-Fradley, K;
Croft, SL;
de Souza, W;
Ruiz-Perez, LM;
+3 more...
Urbina, J;
Pacanowska, DG;
Gilbert, IH;
(2003)
Azasterols as inhibitors of sterol 24-methyltransferase in leishmania species and Trypanosoma cruzi.
Journal of medicinal chemistry, 46 (22).
pp. 4714-4727.
ISSN 0022-2623
DOI: https://doi.org/10.1021/jm021114j
Full text not available from this repository.
2002
Adagu, IS;
Nolder, D;
Warhurst, DC;
Rossignol, JF;
(2002)
In vitro activity of nitazoxanide and related compounds against isolates of Giardia intestinalis, Entamoeba histolytica and Trichomonas vaginalis.
The Journal of antimicrobial chemotherapy, 49 (1).
pp. 103-11.
ISSN 0305-7453
DOI: https://doi.org/10.1093/jac/49.1.103
Full text not available from this repository.
2001
Barlow, SM;
Sullivan, FM;
Lines, J;
(2001)
Risk assessment of the use of deltamethrin on bednets for the prevention of malaria.
Food and chemical toxicology, 39 (5).
pp. 407-422.
ISSN 0278-6915
DOI: https://doi.org/10.1016/S0278-6915(00)00152-6
Full text not available from this repository.
Blackwell, JM;
Goswami, T;
Evans, CA;
Sibthorpe, D;
Papo, N;
White, JK;
Searle, S;
Miller, EN;
Peacock, CS;
Mohammed, H;
+1 more...
Ibrahim, M;
(2001)
SLC11A1 (formerly NRAMP1) and disease resistance.
Cellular microbiology, 3 (12).
pp. 773-84.
ISSN 1462-5814
DOI: https://doi.org/10.1046/j.1462-5822.2001.00150.x
Full text not available from this repository.
Kelly, JM;
Quack, G;
Miles, MM;
(2001)
In vitro and in vivo activities of aminoadamantane and aminoalkylcyclohexane derivatives against Trypanosoma brucei.
Antimicrobial agents and chemotherapy, 45 (5).
pp. 1360-6.
ISSN 0066-4804
DOI: https://doi.org/10.1128/AAC.45.5.1360-1366.2001
Full text not available from this repository.
Martin, MB;
Grimley, JS;
Lewis, JC;
Heath, HT;
Bailey, BN;
Kendrick, H;
Yardley, V;
Caldera, A;
Lira, R;
Urbina, JA;
+4 more...
Moreno, SNJ;
Docampo, R;
Croft, SL;
Oldfield, E;
(2001)
Bisphosphonates inhibit the growth of Trypanosoma brucei, Trypanosoma cruzi, Leishmania donovani, Toxoplasma gondii, and Plasmodium falciparum: A potential route to chemotherapy.
Journal of medicinal chemistry, 44 (6).
pp. 909-16.
ISSN 0022-2623
https://researchonline.lshtm.ac.uk/id/eprint/16563
Full text not available from this repository.
Ohkanda, J;
Lockman, JW;
Yokoyama, K;
Gelb, MH;
Croft, SL;
Kendrick, H;
Harrell, MI;
Feagin, JE;
Blaskovich, MA;
Sebti, SM;
+1 more...
Hamilton, AD;
(2001)
Peptidomimetic inhibitors of protein farnesyltransferase show potent antimalarial activity.
Bioorganic & medicinal chemistry letters, 11 (6).
pp. 761-764.
ISSN 0960-894X
DOI: https://doi.org/10.1016/S0960-894X(01)00055-5
Full text not available from this repository.
Salmon-Chemin, L;
Buisine, E;
Yardley, V;
Kohler, S;
Debreu, MA;
Landry, V;
Sergheraert, C;
Croft, SL;
Krauth-Siegel, RL;
Davioud-Charvet, E;
(2001)
2-and 3-substituted 1,4-naphthoquinone derivatives as subversive substrates of trypanothione reductase and lipoamide dehydrogenase from Trypanosoma cruzi: Synthesis and correlation between redox cycling activities and in vitro cytotoxicity.
Journal of medicinal chemistry, 44 (4).
pp. 548-65.
ISSN 0022-2623
https://researchonline.lshtm.ac.uk/id/eprint/16559
Full text not available from this repository.
Wright, CW;
Addae-Kyereme, J;
Breen, AG;
Brown, JE;
Cox, MF;
Croft, SL;
Gokcek, Y;
Kendrick, H;
Phillips, RM;
Pollet, PL;
(2001)
Synthesis and evaluation of cryptolepine analogues for their potential as new antimalarial agents.
Journal of medicinal chemistry, 44 (19).
pp. 3187-94.
ISSN 0022-2623
https://researchonline.lshtm.ac.uk/id/eprint/16568
Full text not available from this repository.
Wyrsta, MD;
Cogen, AL;
Deming, TJ;
(2001)
A parallel synthetic approach for the analysis of membrane interactive copolypeptides.
Journal of the American Chemical Society, 123 (51).
pp. 12919-20.
ISSN 0002-7863
DOI: https://doi.org/10.1021/ja017307y
Full text not available from this repository.