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Jump to: 2009 | 2008 | 2007 | 2006 | 2005 | 2004 | 2003 | 2002 | 2001
Number of items: 24.

2009

Cogen, AL; Yamasaki, K; Sanchez, KM; Dorschner, RA; Lai, Y; MacLeod, DT; Torpey, JW; Otto, M; Nizet, V; Kim, JE; +1 more... Gallo, RL; (2009) Selective antimicrobial action is provided by phenol-soluble modulins derived from Staphylococcus epidermidis, a normal resident of the skin. The Journal of investigative dermatology, 130 (1). pp. 192-200. ISSN 0022-202X DOI: https://doi.org/10.1038/jid.2009.243 Full text not available from this repository.

2008

Musonda, CC; Yardley, V; de Souza, RCC; Ncokazi, K; Egan, TJ; Chibale, K; (2008) Antiplasmodial, beta-haematin inhibition, antitrypanosomal and cytotoxic activity in vitro of novel 4-aminoquinoline 2-imidazolines. Organic & biomolecular chemistry, 6 (23). pp. 4446-4451. ISSN 1477-0520 DOI: https://doi.org/10.1039/b813007h Full text not available from this repository.

2007

Blackie, MAL; Beagley, P; Croft, SL; Kendrick, H; Moss, JR; Chibale, K; (2007) Metallocene-based antimalarials: An exploration into the influence of the ferrocenyl moiety on in vitro antimalarial activity in chloroquine-sensitive and chloroquine-resistant strains of Plasmodium falciparum. Bioorganic & medicinal chemistry, 15 (20). pp. 6510-6516. ISSN 0968-0896 DOI: https://doi.org/10.1016/j.bmc.2007.07.012 Full text not available from this repository.

Khrizman, A; Moulthrop, JS; Little, S; Wharton, H; Yardley, V; Moyna, G; (2007) Synthesis and in vitro protozoocidal activity of diazabicyclic benzotropolone derivatives. Bioorganic & medicinal chemistry letters, 17 (15). pp. 4183-4186. ISSN 0960-894X DOI: https://doi.org/10.1016/j.bmcl.2007.05.044 Full text not available from this repository.

Musonda, CC; Little, S; Yardley, V; Chibale, K; (2007) Application of multicomponent reactions to antimalarial drug discovery. Part 3: Discovery of aminoxazole 4-aminoquinolines with potent antiplasmodial activity in vitro. Bioorganic & medicinal chemistry letters, 17 (17). pp. 4733-4736. ISSN 0960-894X DOI: https://doi.org/10.1016/j.bmcl.2007.06.070 Full text not available from this repository.

Too, K; Brown, DM; Bongard, E; Yardley, V; Vivas, L; Loakes, D; (2007) Anti-malarial activity of N-6-modified purine analogues. Bioorganic & medicinal chemistry, 15 (16). pp. 5551-5562. ISSN 0968-0896 DOI: https://doi.org/10.1016/j.bmc.2007.05.038 Full text not available from this repository.

van Wyk, AWW; Lobb, KA; Caira, MR; Hoppe, HC; Davies-Coleman, MT; (2007) Transformations of Manool. Tri- and Tetracyclic Norditerpenoids with in Vitro Activity against Plasmodium falciparum. Journal of natural products, 70 (8). pp. 1253-1258. ISSN 0163-3864 DOI: https://doi.org/10.1021/np0701071 Full text not available from this repository.

2006

Hudock, MP; Sanz-Rodriguez, CE; Song, YC; Chan, JMW; Zhang, YH; Odeh, S; Kosztowski, T; Leon-Rossell, A; Concepcion, JL; Yardley, V; +3 more... Croft, SL; Urbina, JA; Oldfield, E; (2006) Inhibition of Trypanosoma cruzi hexokinase by bisphosphonates. Journal of medicinal chemistry, 49 (1). pp. 215-223. ISSN 0022-2623 DOI: https://doi.org/10.1021/jm0582625 Full text not available from this repository.

2005

Lorente, SO; Jimenez, CJ; Gros, L; Yardley, V; de Luca-Fradley, K; Croft, SL; Urbina, JA; Ruiz-Perez, LM; Pacanowska, DG; Gilbert, IH; (2005) Preparation of transition-state analogues of sterol 24-methyl transferase as potential anti-parasities. Bioorganic & medicinal chemistry, 13 (18). pp. 5435-5453. ISSN 0968-0896 DOI: https://doi.org/10.1016/j.bmc.2005.06.012 Full text not available from this repository.

2004

Bhakoo, A; Raynes, JG; Heal, JR; Keller, M; Miller, AD; (2004) De-novo design of complementary (antisense) peptide mini-receptor inhibitor of interleukin 18 (IL-18). Molecular immunology, 41 (12). pp. 1217-1224. ISSN 0161-5890 DOI: https://doi.org/10.1016/j.molimm.2004.05.011 Full text not available from this repository.

Ghosh, S; Chan, JMW; Lea, CR; Meints, GA; Lewis, JC; Tovian, ZS; Flessner, RM; Loftus, TC; Bruchhaus, I; Kendrick, H; +5 more... Croft, SL; Kemp, RG; Kobayashi, S; Nozaki, T; Oldfield, E; (2004) Effects of bisphosphonates on the growth of Entamoeba histolytica and Plasmodium species in vitro and in vivo. Journal of medicinal chemistry, 47 (1). pp. 175-187. ISSN 0022-2623 DOI: https://doi.org/10.1021/jm030084x Full text not available from this repository.

Mantyla, A; Garnier, T; Rautio, R; Nevalainen, T; Vepsalainen, J; Koskinen, A; Croft, SL; Jarvinen, T; (2004) Synthesis, in vitro evaluation, and antileishmanial activity of water-soluble prodrugs of buparvaquone. Journal of medicinal chemistry, 47 (1). pp. 188-195. ISSN 0022-2623 DOI: https://doi.org/10.1021/jm030868a Full text not available from this repository.

2003

Chauviere, G; Bouteille, B; Enanga, B; de Albuquerque, C; Croft, SL; Dumas, M; Perie, J; (2003) Synthesis and biological activity of nitro heterocycles analogous to megazol, a trypanocidal lead. Journal of medicinal chemistry, 46 (3). pp. 427-440. ISSN 0022-2623 DOI: https://doi.org/10.1021/jm021030a Full text not available from this repository.

Magaraci, F; Jimenez, CJ; Rodrigues, C; Rodrigues, JCF; Braga, MV; Yardley, V; de Luca-Fradley, K; Croft, SL; de Souza, W; Ruiz-Perez, LM; +3 more... Urbina, J; Pacanowska, DG; Gilbert, IH; (2003) Azasterols as inhibitors of sterol 24-methyltransferase in leishmania species and Trypanosoma cruzi. Journal of medicinal chemistry, 46 (22). pp. 4714-4727. ISSN 0022-2623 DOI: https://doi.org/10.1021/jm021114j Full text not available from this repository.

2002

Jiang, S; Borthwick, NJ; Morrison, P; Gao, GF; Steward, MW; (2002) Virus-specific CTL responses induced by an H-2K(d)-restricted, motif-negative 15-mer peptide from the fusion protein of respiratory syncytial virus. The Journal of general virology, 83 (Pt 2). pp. 429-38. ISSN 0022-1317 http://researchonline.lshtm.ac.uk/id/eprint/17357 Full text not available from this repository.

Jung, MK; Lee, K; Kendrick, H; Robinson, BL; Croft, SL; (2002) Synthesis, stability, and antimalarial activity of new hydrolytically stable and water-soluble (+)-deoxoartelinic acid. Journal of medicinal chemistry, 45 (22). pp. 4940-4. ISSN 0022-2623 DOI: https://doi.org/10.1021/jm020244p Full text not available from this repository.

2001

Chibale, K; Haupt, H; Kendrick, H; Yardley, V; Saravanamuthu, A; Fairlamb, AH; Croft, SL; (2001) Antiprotozoal and cytotoxicity evaluation of sulfonamide and urea analogues of quinacrine. Bioorganic & medicinal chemistry letters, 11 (19). pp. 2655-2657. ISSN 0960-894X DOI: https://doi.org/10.1016/S0960-894X(01)00528-5 Full text not available from this repository.

Daunes, S; D'Silva, C; Kendrick, H; Yardley, V; Croft, SL; (2001) QSAR study on the contribution of log P and E-s to the in vitro antiprotozoal activity of glutathione derivatives. Journal of medicinal chemistry, 44 (18). pp. 2976-83. ISSN 0022-2623 http://researchonline.lshtm.ac.uk/id/eprint/16567 Full text not available from this repository.

Murray, PJ; Kranz, M; Ladlow, M; Taylor, S; Berst, F; Holmes, AB; Keavey, KN; Jaxa-Chamiec, A; Seale, PW; Stead, P; +4 more... Upton, RJ; Croft, SL; Clegg, W; Elsegood, MRJ; (2001) The synthesis of cyclic tetrapeptoid analogues of the antiprotozoal natural product apicidin. Bioorganic & medicinal chemistry letters, 11 (6). pp. 773-776. ISSN 0960-894X DOI: https://doi.org/10.1016/S0960-894X(01)00049-X Full text not available from this repository.

Ohkanda, J; Lockman, JW; Yokoyama, K; Gelb, MH; Croft, SL; Kendrick, H; Harrell, MI; Feagin, JE; Blaskovich, MA; Sebti, SM; +1 more... Hamilton, AD; (2001) Peptidomimetic inhibitors of protein farnesyltransferase show potent antimalarial activity. Bioorganic & medicinal chemistry letters, 11 (6). pp. 761-764. ISSN 0960-894X DOI: https://doi.org/10.1016/S0960-894X(01)00055-5 Full text not available from this repository.

Ren, HY; Grady, S; Gamenara, D; Heinzen, H; Moyna, P; Croft, SL; Kendrick, H; Yardley, V; Moyna, G; (2001) Design, synthesis, and biological evaluation of a series of simple and novel potential antimalarial compounds. Bioorganic & medicinal chemistry letters, 11 (14). pp. 1851-1854. ISSN 0960-894X DOI: https://doi.org/10.1016/S0960-894X(01)00308-0 Full text not available from this repository.

Salmon-Chemin, L; Buisine, E; Yardley, V; Kohler, S; Debreu, MA; Landry, V; Sergheraert, C; Croft, SL; Krauth-Siegel, RL; Davioud-Charvet, E; (2001) 2-and 3-substituted 1,4-naphthoquinone derivatives as subversive substrates of trypanothione reductase and lipoamide dehydrogenase from Trypanosoma cruzi: Synthesis and correlation between redox cycling activities and in vitro cytotoxicity. Journal of medicinal chemistry, 44 (4). pp. 548-65. ISSN 0022-2623 http://researchonline.lshtm.ac.uk/id/eprint/16559 Full text not available from this repository.

Wright, CW; Addae-Kyereme, J; Breen, AG; Brown, JE; Cox, MF; Croft, SL; Gokcek, Y; Kendrick, H; Phillips, RM; Pollet, PL; (2001) Synthesis and evaluation of cryptolepine analogues for their potential as new antimalarial agents. Journal of medicinal chemistry, 44 (19). pp. 3187-94. ISSN 0022-2623 http://researchonline.lshtm.ac.uk/id/eprint/16568 Full text not available from this repository.

Wyrsta, MD; Cogen, AL; Deming, TJ; (2001) A parallel synthetic approach for the analysis of membrane interactive copolypeptides. Journal of the American Chemical Society, 123 (51). pp. 12919-20. ISSN 0002-7863 DOI: https://doi.org/10.1021/ja017307y Full text not available from this repository.

This list was generated on Thu Mar 21 11:12:08 2019 GMT.